The goal of the project is to use microwave technology to synthesise benzocain and evaluate its antibacterial qualities. Benzodiazepines are the best example of anaesthetic agents. According to the protocol, it is made by condensation of amino benzoic acid and HCl with ethanol, a CNS depressant, serving as a solvent. Additional UV spectrum verification of benzocain production. Additional proof for synthesised benzocain was supplied by FTIR. The fluorescence behaviour of the synthesised benzocain was examined. Benzocaines antibacterial activity against Escherichia coli and Staphylococcus aureus has been verified. In general, green chemistry principles are used in the synthesis of benzocaine, and the use of ethanol assures its safety. The utilization of microwave synthesis for the synthesis of benzocaine and a possible antibacterial drug results in a reduction of both time and cost. Here, we report a microwave-assisted benzocaine synthesis that makes use of easily accessible precursors and microwave irradiation as the heating medium. The efficacy and adaptability of the microwaveassisted method were demonstrated when the reaction was tuned to provide high yields under moderate circumstances. Using spectroscopic methods, the synthesised benzocaine was characterised, confirming its authenticity and purity.